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December 8, 2025BloodOpen Access

Bexobrutideg (NX-5948), a novel Bruton's tyrosine kinase (BTK) degrader, shows high clinical activity and tolerable safety in patients with Waldenström macroglobulinemia: Updated results from an ongoing Phase 1a/b study

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Authors

NSNirav N. ShahKLKim LintonDEDima El‐Sharkawi

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Overview

Updated analysis reveals high overall response rates in patients with Waldenström macroglobulinemia, suggesting Bexobrutideg's potential in B-cell malignancies.

Key Points

  • Overall response rate reached 85.0% in patients with Waldenström macroglobulinemia, showing significant clinical activity.
  • Patients demonstrated a median IgM reduction of 79.6%, indicating effective treatment response.
  • Analysis from an ongoing Phase 1a/b trial assessed safety and preliminary efficacy of Bexobrutideg in B-cell malignancies.
  • Findings highlight Bexobrutideg's tolerability and efficacy, with ongoing expansion in Phase 1b study.

Cite This Study

Shah et al. (2025) studied this question.

synapsesocial.com/papers/69362f5a4fa91c937236db30https://doi.org/10.1182/blood-2025-5359
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